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N-(2-hydroxyethyl)-n-methyl-4-(quinolin-8-yl(1-(thiazol-4-ylmethyl) piperidin-4-ylidene)methyl)benzamide, method for preparing and applying it for treating pain, anxiety and depression. RU patent 2454414.

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to N-(2-hydroxyethyl)-N-methyl-4-(quinolin-8-yl(1-(thiazol-4-ylmethyl)-piperidin-4-ylidene)methyl)benzamide, and/or their mixture, as well as to applying it in a pharmaceutical composition, a method of treating to be applied for treating pain, anxiety, depression, worried depression or Parkinson's disease. Also, the invention refers to methods for preparing N-(2-hydroxyethyl)-N-methyl-4-(quinolin-8-yl(1-(thiazol-4-ylmethyl)-piperidin-4-ylidene)methyl)benzamide and its intermediate compounds. .

EFFECT: developing the method of treating to be applied for treating pain, anxiety, depression, worried depression or Parkinson's disease.

12 cl, 1 ex

IPC classes for russian patent N-(2-hydroxyethyl)-n-methyl-4-(quinolin-8-yl(1-(thiazol-4-ylmethyl) piperidin-4-ylidene)methyl)benzamide, method for preparing and applying it for treating pain, anxiety and depression. RU patent 2454414. (RU 2454414):

C07D417/14 - containing three or more hetero rings

C07D401/08 - linked by a carbon chain containing alicyclic rings

A61P25/24 - Antidepressants

A61P25/22 - Anxiolytics

A61P25/16 - Anti-Parkinson drugs

A61P25/04 - Centrally acting analgesics, e.g. opioids

A61K31/4709 -

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