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Diarylmetyhylpyperazine derivatives, their obtaining and application. RU patent 2404172.

Diarylmetyhylpyperazine derivatives, their obtaining and application. RU patent 2404172.

FIELD: medicine.

SUBSTANCE: there are described compound of formula, its pharmaceutically acceptable salt or their mixture, enentiomerically pure 4-{(R)-(3-aminophenyl)[4-(4-fluorobenzyl)pyperazin-1-yl]-N,N-diethylbenzamide or its pharmaceutically acceptable salt. Also described are method of anxiety therapy, method of pain therapy and method of depression therapy in animal.

EFFECT: compounds are of use in therapy, in particular for elimination of pain, depression and anxiety.

5 cl, 1 tbl, 9 ex

 


 

IPC classes for russian patent Diarylmetyhylpyperazine derivatives, their obtaining and application. RU patent 2404172. (RU 2404172):

C07D295/155 -
A61P25/24 - Antidepressants
A61P25/22 - Anxiolytics
A61P25/04 - Centrally acting analgesics, e.g. opioids
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